SCHEMBL1702937

SCHEMBL1702937

Nc1n[nH]c2nccc(-c3ccc(NC(=O)Nc4ccc(F)c(C(F)(F)F)c4)cc3)c12

nearest known ligand 0.75

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.75
KIT P10721 12/20 0.67
FLT3 P36888 12/20 0.67
CSF1R P07333 6/20 0.67
LCK P06239 5/20 0.67
LYN P07948 5/20 0.67
SRC P12931 5/20 0.67
FLT4 P35916 5/20 0.67
BLK P51451 5/20 0.67
FLT1 P17948 5/20 0.67
ABL1 P00519 3/20 0.67
RIPK1 Q13546 2/20 0.64
FYN P06241 5/20 0.57
NTRK1 P04629 1/20 0.55
IKBKE Q14164 1/20 0.55
CDK19 Q9BWU1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2236868 0.89 KDR (0.60) KDRKITFLT3CSF1RLCK
SCHEMBL1703109 0.86 KDR (0.74) KDRKITFLT3CSF1RLCK
SCHEMBL1703083 0.86 KDR (0.74) KDRKITFLT3CSF1RLCK
SCHEMBL1703063 0.86 KDR (0.77) KDRKITFLT3CSF1RLCK
SCHEMBL1702788 0.85 KDR (0.76) KDRKITFLT3CSF1RLCK
SCHEMBL425326 0.84 KDR (0.75) KDRKITFLT3CSF1RLCK
SCHEMBL1702977 0.84 KDR (0.75) KDRKITFLT3CSF1RLCK
SCHEMBL420525 0.84 KDR (0.63) KDRKITFLT3CSF1RLCK
SCHEMBL422215 0.83 KDR (0.62) KDRKITFLT3CSF1RLCK
SCHEMBL1702906 0.83 KDR (0.72) KDRKITFLT3CSF1RLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807424-B1 NOVEL KINASE INHIBITORS ABBOTT LAB (US) 2012-04-18 EP claimed
EP-1807424-A2 NOVEL KINASE INHIBITORS ABBOTT LABORATORIES (US) 2007-07-18 EP claimed
US-20060178378-A1 Novel kinase inhibitors ABBVIE INC. 2006-08-10 US claimed
WO-2006050109-A2 NOVEL KINASE INHIBITORS ABBOTT LABORATORIES (US) 2006-05-11 WO claimed
EP-1807424-B1 NOVEL KINASE INHIBITORS ABBOTT LAB (US) 2012-04-18 EP disclosed
US-7812166-B2 Kinase inhibitors ABBOTT LABORATORIES (US) 2010-10-12 US disclosed
US-20060178378-A1 Novel kinase inhibitors ABBVIE INC. 2006-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060178378-A1 Novel kinase inhibitors ABL1, MAP3K19, MAP3K20 KDR 434/4885KIT 426/4885FLT3 79/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.