SCHEMBL17044153

SCHEMBL17044153

CC(Cc1ccc2c(c1)CN(C)CC2c1ccc2ccoc2c1)N1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 20/20 0.58
SLC6A3 Q01959 15/20 0.58
SLC6A2 P23975 14/20 0.58
CYP2D6 P10635 1/20 0.44
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313152 0.85 SLC6A4 (0.62) SLC6A4SLC6A3SLC6A2CYP2D6KCNH2
SCHEMBL4305751 0.81 SLC6A4 (0.69) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL4308682 0.80 SLC6A4 (0.64) SLC6A4SLC6A3SLC6A2HRH3
SCHEMBL17044152 0.80 SLC6A4 (0.58) SLC6A4SLC6A3SLC6A2CYP2D6KCNH2
SCHEMBL4303606 0.80 SLC6A4 (0.69) SLC6A4SLC6A3SLC6A2CYP2D6KCNH2
SCHEMBL4312426 0.80 SLC6A4 (0.66) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL4306331 0.80 SLC6A4 (0.66) SLC6A4SLC6A3SLC6A2CYP2D6KCNH2
SCHEMBL4308404 0.79 SLC6A4 (0.62) SLC6A4SLC6A3SLC6A2HRH3
SCHEMBL4309477 0.79 SLC6A4 (0.61) SLC6A4SLC6A3SLC6A2CYP2D6KCNH2
SCHEMBL4303961 0.77 SLC6A2 (0.74) SLC6A4SLC6A3SLC6A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778639-B1 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN ALBANY MOLECULAR RES INC (US) 2015-09-02 EP disclosed