SCHEMBL17044359

SCHEMBL17044359

CC1(c2ccccc2)CCN2CCC(C)(c3ccccc3)c3cc(NC(=O)O)cc1c32

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FSHR P23945 9/20 0.41
MMP1 P03956 2/20 0.41
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
TSHR P16473 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EPHX2 P34913 3/20 0.37
ADAM17 P78536 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ADRB2 P07550 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3160570 1.00 FSHR (0.41) FSHRMMP1MMP2MMP9TSHR
SCHEMBL2388862 1.00 FSHR (0.41) FSHRMMP1MMP2MMP9TSHR
SCHEMBL11973791 0.91 FSHR (0.41) FSHRMMP1MMP2MMP9TSHR
SCHEMBL11973331 0.91 FSHR (0.41) FSHRMMP1MMP2MMP9TSHR
SCHEMBL17054382 0.90 FSHR (0.40) FSHRMMP1MMP2MMP9TSHR
SCHEMBL8988202 0.89 FSHR (0.44) FSHRMMP1MMP2MMP9TSHR
SCHEMBL11973796 0.89 TP53 (0.38) TSHR
SCHEMBL2389637 0.89 FSHR (0.44) FSHRMMP1MMP2MMP9TSHR
SCHEMBL2392497 0.89 FSHR (0.44) FSHRMMP1MMP2MMP9TSHR
SCHEMBL2392758 0.89 FSHR (0.41) FSHRMMP1MMP2MMP9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2294069-B1 THERAPEUTICALLY USEFUL SUBSTITUTED HYDROPYRIDO[3,2,1-IJ]QUINOLINE COMPOUNDS ALLERGAN INC (US) 2015-09-02 EP disclosed