SCHEMBL1705074

SCHEMBL1705074

CC(C)N1CCN(c2ccc(Nc3nc(N4CCC[C@@H](Nc5ccccc5)C4)ccc3C(N)=O)cc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTK Q06187 17/20 0.57
KCNH2 Q12809 2/20 0.57
JAK3 P52333 7/20 0.47
LCK P06239 4/20 0.47
EGFR P00533 1/20 0.47
SYK P43405 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL893881 0.90 BTK (0.58) BTKKCNH2JAK3LCKEGFR
SCHEMBL893880 0.90 BTK (0.58) BTKKCNH2JAK3LCKEGFR
SCHEMBL894610 0.81 BTK (0.61) BTKKCNH2JAK3LCKEGFR
SCHEMBL894964 0.78 BTK (0.59) BTKKCNH2JAK3LCKEGFR
SCHEMBL895137 0.78 BTK (0.61) BTKKCNH2JAK3LCKEGFR
SCHEMBL893992 0.77 BTK (0.61) BTKKCNH2JAK3LCKEGFR
SCHEMBL893995 0.77 BTK (0.61) BTKKCNH2JAK3LCKEGFR
SCHEMBL10210795 0.75 BTK (0.54) BTKKCNH2JAK3LCKEGFR
SCHEMBL1705497 0.75 BTK (0.54) BTKKCNH2JAK3LCKEGFR
SCHEMBL10211523 0.75 BTK (0.52) BTKKCNH2JAK3LCKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440204-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS Bristol-Myers Squibb Company (US) 2012-04-18 EP disclosed
WO-2010144647-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-12-16 WO disclosed