SCHEMBL17059333

SCHEMBL17059333

C=CCc1cc(Nc2nccc(-c3cnc4ccccc4c3)n2)c(OC)cc1N1CC[C@@H](N(C)C)C1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.53
INSR P06213 2/20 0.43
IGF1R P08069 2/20 0.43
KCNH2 Q12809 1/20 0.43
ALK Q9UM73 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18369607 0.87 EGFR (0.51) EGFRINSRIGF1RKCNH2ALK
SCHEMBL20578395 0.85 EGFR (0.73) EGFRINSRIGF1RKCNH2
SCHEMBL18359243 0.85 EGFR (0.73) EGFRINSRIGF1RKCNH2
SCHEMBL17059329 0.84 EGFR (0.50) EGFRINSRIGF1RKCNH2ALK
SCHEMBL17059287 0.81 EGFR (0.80) EGFR
SCHEMBL17059313 0.81 EGFR (0.55) EGFRINSRIGF1R
SCHEMBL17059293 0.79 EGFR (0.78) EGFRINSRIGF1RKCNH2
SCHEMBL17059332 0.77 EGFR (0.53) EGFRINSRIGF1RKCNH2
SCHEMBL28383483 0.72 EGFR (0.67) EGFRINSRIGF1RKCNH2ALK
SCHEMBL17059292 0.72 EGFR (0.78) EGFRIGF1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015127872-A1 2,4-DISUBSTITUTED PHENYLENE-1,5-DIAMINE DERIVATIVES AND APPLICATIONS THEREOF, AND PHARMACEUTICAL COMPOSITIONS AND PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS PREPARED THEREFROM 上海海雁医药科技有限公司 2015-09-03 WO disclosed