SCHEMBL17065178

SCHEMBL17065178

N#Cc1cccc(-c2ccncn2)c1-c1ccncn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.49
UCHL1 P09936 1/20 0.41
HTT P42858 1/20 0.40
GSK3B P49841 2/20 0.36
CYP2D6 P10635 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NFATC1 O95644 1/20 0.35
DYRK1A Q13627 1/20 0.35
PDK2 Q15119 1/20 0.35
NISCH Q9Y2I1 1/20 0.34
ADORA2B P29275 1/20 0.34
EZH2 Q15910 1/20 0.34
CCNT1 O60563 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16797340 0.87 GRM5 (0.42) GRM5UCHL1GSK3BCYP2D6MEN1
SCHEMBL18151343 0.87 GRM5 (0.42) GRM5UCHL1HTTGSK3BCYP2D6
SCHEMBL27852673 0.86 GRM5 (0.44) GRM5UCHL1HTTGSK3BCYP2D6
SCHEMBL30485537 0.86 GRM5 (0.44) GRM5UCHL1HTTGSK3BCYP2D6
SCHEMBL18151571 0.86 GRM5 (0.41) GRM5UCHL1GSK3BCYP2D6MEN1
SCHEMBL30893416 0.85 GRM5 (0.44) GRM5UCHL1HTTGSK3BCYP2D6
SCHEMBL18151348 0.85 GRM5 (0.43) GRM5UCHL1HTTGSK3BCYP2D6
SCHEMBL16797343 0.85 LRRK2 (0.44) GRM5UCHL1GSK3BCYP2D6MEN1
SCHEMBL30401803 0.85 GRM5 (0.40) GRM5UCHL1HTTGSK3BCYP2D6
SCHEMBL18151573 0.84 GRM5 (0.42) GRM5UCHL1HTTGSK3BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015134536-A1 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC. (US) 2015-09-11 WO disclosed