SCHEMBL17065331

SCHEMBL17065331

CC(C)(C)[Si](OCC1CN(C(=O)O)CC(CCc2ccccc2N)O1)(c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 3/20 0.35
CYP3A4 P08684 2/20 0.31
PSMB5 P28074 1/20 0.30
SIRT2 Q8IXJ6 1/20 0.30
SIRT1 Q96EB6 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19179494 1.00 SMYD2 (0.35) SMYD2CYP3A4PSMB5SIRT2SIRT1
SCHEMBL19181572 0.89 SIRT2 (0.31) SIRT2SIRT1
SCHEMBL17065329 0.84 SMYD2 (0.37) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL16834440 0.84 SMYD2 (0.33) SMYD2CYP3A4
SCHEMBL17065394 0.83 SMYD2 (0.36) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL17065348 0.83 SMYD2 (0.38) SMYD2CYP3A4PSMB5HTTSMN1; SMN2
SCHEMBL19180508 0.82 SMYD2 (0.37) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL19181577 0.80 SMYD2 (0.37) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL19181556 0.79 SMYD2 (0.37) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL17065382 0.78 KDM4E (0.36) SMYD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3113780-A1 HIV PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-01-11 EP disclosed
WO-2015134366-A1 HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-09-11 WO disclosed