SCHEMBL17066009

SCHEMBL17066009

O=C(Nc1cn2cc(B(O)O)ccc2n1)C1CC1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 10/20 0.53
MAP4K1 Q92918 6/20 0.50
ABL1 P00519 5/20 0.48
HPGD P15428 1/20 0.45
KDR P35968 3/20 0.43
AURKA O14965 1/20 0.43
PDGFRB P09619 1/20 0.43
KIT P10721 1/20 0.43
FLT1 P17948 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1259693 0.82 LRRK2 (0.56) LRRK2MAP4K1ABL1HPGDKDR
SCHEMBL3145952 0.82 PIK3CA (0.50) HPGDKDR
SCHEMBL24305376 0.81 LRRK2 (0.55) LRRK2MAP4K1ABL1HPGDKDR
SCHEMBL17065938 0.81 MAP3K5 (0.56) LRRK2MAP4K1ABL1HPGDKDR
SCHEMBL1258121 0.74 KDR (0.55) LRRK2MAP4K1ABL1KDRAURKA
SCHEMBL17066024 0.73 LRRK2 (0.46) LRRK2MAP4K1ABL1KDRAURKA
SCHEMBL24296473 0.73 LRRK2 (0.56) LRRK2MAP4K1ABL1HPGDKDR
SCHEMBL22380353 0.73 LRRK2 (0.55) LRRK2MAP4K1ABL1
SCHEMBL22380367 0.73 LRRK2 (0.77) LRRK2MAP4K1ABL1
SCHEMBL31557493 0.72 JAK1 (0.57) LRRK2HPGDKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015134171-A1 HETEROARYLAMIDE INHIBITORS OF TBK1 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-09-11 WO disclosed