SCHEMBL1708386

SCHEMBL1708386

CCOc1nc2ccccc2n1-c1cccc2c1OC[C@@H]2N(C(=O)C(F)(F)F)c1ccc2c(c1)OC(C)[C@H]2OC(C)=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708331 1.00
SCHEMBL1708327 0.93
SCHEMBL1708144 0.93
SCHEMBL1708019 0.92
SCHEMBL1707978 0.91 CHEK1 (0.30)
SCHEMBL1708025 0.91 CHEK1 (0.30)
SCHEMBL1708118 0.90 TSHR (0.32)
SCHEMBL1708050 0.90 TSHR (0.32)
SCHEMBL1707936 0.90 TSHR (0.32)
SCHEMBL1708380 0.89

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed