SCHEMBL17089991

SCHEMBL17089991

C[C@@H]1CN(c2ccc(NC[C@H]3CC[C@H](NS(=O)(=O)C(C)(C)C)CC3)cn2)C[C@H](C)O1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.39
KCNH2 Q12809 1/20 0.39
SMO Q99835 2/20 0.37
PGR P06401 1/20 0.37
GPR183 P32249 1/20 0.37
MET P08581 1/20 0.36
NPY5R Q15761 1/20 0.35
LRRK2 Q5S007 1/20 0.35
BCL6 P41182 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
AOC3 Q16853 1/20 0.34
KMT2A Q03164 1/20 0.33
DYRK1A Q13627 2/20 0.33
CLK2 P49760 1/20 0.33
CLK3 P49761 1/20 0.33
WNT1 P04628 1/20 0.33
ADRA1A P35348 1/20 0.33
KDM1A O60341 1/20 0.33
CRHR1 P34998 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565822 1.00 BTK (0.39) BTKKCNH2SMOPGRGPR183
SCHEMBL13565556 0.89 SYK (0.40) BTKKCNH2METKMT2AKDM1A
SCHEMBL11935391 0.87 BTK (0.37) BTKKCNH2SMOPGRGPR183
SCHEMBL13439104 0.87 BTK (0.37) BTKKCNH2SMOPGRGPR183
SCHEMBL17090150 0.87 BTK (0.37) BTKKCNH2SMOPGRGPR183
SCHEMBL13564738 0.85 MAPT (0.43) LRRK2
SCHEMBL11936149 0.85 MAPT (0.43) LRRK2
SCHEMBL13565140 0.85 MAPT (0.43) LRRK2
SCHEMBL17089987 0.85 MAPT (0.43) LRRK2
SCHEMBL10133762 0.82 NPY5R (0.52) BTKKCNH2SMOPGRGPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed