SCHEMBL17090397

SCHEMBL17090397

CCCC(C)S(=O)(=O)N[C@H]1CC[C@H](CNc2ccc3ncsc3c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 14/20 0.42
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
UBE2M P61081 1/20 0.41
DCUN1D1 Q96GG9 1/20 0.41
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40
RIPK1 Q13546 1/20 0.37
JAK3 P52333 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4D Q08499 1/20 0.37
CHRM5 P08912 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565309 1.00 IRAK4 (0.42) IRAK4TAS1R3TAS1R1UBE2MDCUN1D1
SCHEMBL17090186 0.92 IRAK4 (0.43) IRAK4UBE2MDCUN1D1ALDH1A1PKM
SCHEMBL13565995 0.92 IRAK4 (0.43) IRAK4UBE2MDCUN1D1ALDH1A1PKM
SCHEMBL11936271 0.89 IRAK4 (0.45) IRAK4ALDH1A1PKMRIPK1JAK3
SCHEMBL11935137 0.89 IRAK4 (0.45) IRAK4ALDH1A1PKMRIPK1JAK3
SCHEMBL10114877 0.83 CHRM5 (0.51) IRAK4TAS1R3TAS1R1UBE2MDCUN1D1
SCHEMBL14424373 0.83 CHRM5 (0.51) IRAK4TAS1R3TAS1R1UBE2MDCUN1D1
SCHEMBL17089965 0.81 IRAK4 (0.47) IRAK4ALDH1A1PKMJAK3
SCHEMBL13565395 0.81 IRAK4 (0.47) IRAK4ALDH1A1PKMJAK3
SCHEMBL17090421 0.81 RIPK2 (0.41) IRAK4ALDH1A1RIPK1CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed