SCHEMBL17101374

SCHEMBL17101374

CCc1nc(C(=O)N2CCCC3(CCN(Cc4cccc(CCOCCC(=O)N(CCNCCc5ccc(O)c6c5OCC(=O)N6)C5CCCC5)c4Cl)CO3)C2)cs1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 9/20 0.46
CHRM2 P08172 7/20 0.38
CHRM3 P20309 7/20 0.38
ADRB2 P07550 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1246208 0.95 SMYD2 (0.47) SMYD2CHRM2CHRM3ADRB2
Sulfuric Acid SCHEMBL1245244 0.93 SMYD2 (0.45) SMYD2CHRM2CHRM3ADRB2
Trifluoroacetic Acid SCHEMBL6525747 0.92 SMYD2 (0.46) SMYD2CHRM2CHRM3ADRB2
SCHEMBL12847000 0.88 SMYD2 (0.47) SMYD2CHRM2CHRM3ADRB2
SCHEMBL12846797 0.87 CHRM2 (0.45) SMYD2CHRM2CHRM3ADRB2
SCHEMBL14576249 0.87 SMYD2 (0.50) SMYD2CHRM2CHRM3ADRB2
SCHEMBL12847130 0.86 CHRM3 (0.44) SMYD2CHRM2CHRM3ADRB2
SCHEMBL12846800 0.86 CHRM2 (0.44) SMYD2CHRM2CHRM3ADRB2
Trifluoroacetic Acid SCHEMBL6524593 0.85 SMYD2 (0.46) SMYD2CHRM2CHRM3ADRB2
SCHEMBL12847100 0.85 CHRM2 (0.44) SMYD2CHRM2CHRM3ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3119752-A1 CHEMICAL COMPOUNDS Astrazeneca AB (SE) 2017-01-25 EP disclosed
WO-2015140527-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2015-09-24 WO disclosed