SCHEMBL17102470

SCHEMBL17102470

CNc1[nH]c(=O)ccc1-c1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 9/20 0.51
PDE3A Q14432 9/20 0.51
AURKB Q96GD4 1/20 0.41
INCENP Q9NQS7 1/20 0.41
GSK3B P49841 2/20 0.39
PARP10 Q53GL7 1/20 0.39
PARP11 Q9NR21 1/20 0.39
PDE10A Q9Y233 3/20 0.38
KDM4E B2RXH2 1/20 0.38
PDE5A O76074 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
PTGS1 P23219 1/20 0.38
PDE4A P27815 1/20 0.38
CYP2C19 P33261 1/20 0.38
BLM P54132 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11117779 0.77 PDE3B (0.56) PDE3BPDE3AAURKBINCENPGSK3B
SCHEMBL11237674 0.72 PDE3B (0.48) PDE3BPDE3AAURKBINCENPGSK3B
SCHEMBL11238085 0.72 PDE3B (0.48) PDE3BPDE3AAURKBINCENPGSK3B
SCHEMBL11109882 0.72 PDE3B (0.55) PDE3BPDE3AAURKBINCENPGSK3B
SCHEMBL11225665 0.70 PDE3B (0.57) PDE3BPDE3AAURKBINCENPGSK3B
SCHEMBL11238852 0.69 GSK3B (0.50) PDE3BPDE3AAURKBINCENPGSK3B
SCHEMBL11226843 0.68 NOTUM (0.67) PDE3BPDE3AGSK3BLMNACDC7
SCHEMBL11243116 0.68 GSK3B (0.51) PDE3BPDE3AAURKBINCENPGSK3B
SCHEMBL26620931 0.67 CA12 (0.35) PDE3BPDE3AKDM4ECYP2C19
SCHEMBL11224039 0.67 PDE3B (0.47) PDE3BPDE3AGSK3BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9145393-B2 Arylpyridinone ITK inhibitors for treating inflammation and cancer CONFLUENCE LIFE SCIENCES, INC. (US) 2015-09-29 US disclosed