SCHEMBL17128683

SCHEMBL17128683

CCCN(CC1CC1)c1cc(C(=O)Nc2ccc(S(=O)(=O)C(CC)C(=O)O)cc2)ncn1

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.76
S1PR3 Q99500 2/20 0.59
S1PR5 Q9H228 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3035013 0.87 S1PR1 (1.00) S1PR1S1PR3S1PR5
SCHEMBL13216786 0.86 S1PR1 (0.88) S1PR1S1PR3S1PR5
SCHEMBL15372630 0.84 S1PR1 (0.80) S1PR1S1PR3S1PR5
SCHEMBL15372608 0.84 S1PR1 (0.82) S1PR1S1PR3S1PR5
SCHEMBL3034983 0.82 S1PR1 (1.00) S1PR1S1PR3S1PR5
SCHEMBL13216771 0.82 S1PR1 (0.85) S1PR1S1PR3S1PR5
SCHEMBL13216802 0.81 S1PR1 (0.88) S1PR1S1PR3S1PR5
SCHEMBL3025823 0.80 S1PR1 (1.00) S1PR1S1PR3S1PR5
SCHEMBL3026901 0.79 S1PR1 (1.00) S1PR1S1PR3
SCHEMBL3025287 0.78 S1PR1 (0.82) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9150519-B2 6-amino-pyrimidine-4-carboxamide derivatives and related compounds which bind to the sphingosine 1-phosphate (S1P) receptor for the treatment of multiple sclerosis MERCK SERONO SA (CH) 2015-10-06 US disclosed