SCHEMBL17147302

SCHEMBL17147302

CCCN1C(=O)CC2(CCN(C)CC2)C1=O

nearest known ligand 0.78

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.78
CHRM3 P20309 1/20 0.78
BDKRB2 P30411 1/20 0.39
CYP19A1 P11511 2/20 0.38
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1043555 0.88 CHRM2 (1.00) CHRM2CHRM3ADRA1AADRA1BL3MBTL1
Bromide SCHEMBL6649504 0.86 CHRM2 (0.97) CHRM2CHRM3ADRA1AADRA1BL3MBTL1
SCHEMBL12787584 0.85 CHRM2 (0.71) CHRM2CHRM3ADRA1AADRA1B
SCHEMBL1043522 0.85 CHRM2 (0.71) CHRM2CHRM3ADRA1AADRA1B
Bromide SCHEMBL194843 0.85 CHRM2 (0.93) CHRM2CHRM3ADRA1AADRA1BL3MBTL1
SCHEMBL1044113 0.85 CHRM2 (0.71) CHRM2CHRM3ADRA1AADRA1B
SCHEMBL1042163 0.81 CHRM2 (0.65) CHRM2CHRM3ADRA1AADRA1BL3MBTL1
SCHEMBL18179697 0.80 CHRM2 (0.69) CHRM2CHRM3ADRA1AADRA1B
SCHEMBL12787585 0.78 CHRM2 (0.65) CHRM2CHRM3BDKRB2ADRA1AADRA1B
SCHEMBL1039704 0.78 CHRM2 (0.65) CHRM2CHRM3BDKRB2ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160310503-A1 Combination Therapies for the Treatment of Alzheimer's Disease and Related Disorders THE GENERAL HOSPITAL CORPORATION 2016-10-27 US disclosed
US-20160310503-A1 Combination Therapies for the Treatment of Alzheimer's Disease and Related Disorders THE GENERAL HOSPITAL CORPORATION 2016-10-27 US disclosed
US-20160271277-A1 Combination Therapies for the Treatment of Alzheimer's Disease and Related Disorders THE GENERAL HOSPITAL CORPORATION 2016-09-22 US disclosed
US-20160166534-A1 Combination Therapies for the Treatment of Alzheimer's Disease and Related Disorders THE GENERAL HOSPITAL CORPORATION 2016-06-16 US disclosed
US-20150283113-A1 COMBINATION THERAPIES FOR THE TREATMENT OF ALZHEIMER'S DISEASE AND RELATED DISORDERS THE GENERAL HOSPITAL CORPORATION 2015-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160166534-A1 Combination Therapies for the Treatment of Alzheimer's Disease and Related Disorders APP, SNCA, MAPT CHRM2 1187/4885CHRM3 1391/4885BDKRB2 2966/4885
US-20160310503-A1 Combination Therapies for the Treatment of Alzheimer's Disease and Related Disorders APP, SNCA, MAPT CHRM2 1187/4885CHRM3 1391/4885BDKRB2 2966/4885
US-20160271277-A1 Combination Therapies for the Treatment of Alzheimer's Disease and Related Disorders APP, SNCA, MAPT CHRM2 1187/4885CHRM3 1391/4885BDKRB2 2966/4885
US-20150283113-A1 COMBINATION THERAPIES FOR THE TREATMENT OF ALZHEIMER'S DISEASE AND RELATED DISORDERS APP, SNCA, MAPT CHRM2 1187/4885CHRM3 1391/4885BDKRB2 2966/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.