SCHEMBL17154283

SCHEMBL17154283

Cc1ccc2c(Oc3ccc(OCCN4CCCCC4)cc3)c(-c3ccc(Br)cc3)sc2c1

nearest known ligand 0.80

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 18/20 0.80
ESR2 Q92731 17/20 0.80
LTA4H P09960 1/20 0.54
PTGS2 P35354 1/20 0.54
ENPP1 P22413 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17154281 0.91 ESR1 (0.85) ESR1ESR2PTGS2
SCHEMBL17154284 0.89 ESR1 (1.00) ESR1ESR2PTGS2
SCHEMBL17155585 0.88 ESR1 (0.76) ESR1ESR2LTA4HPTGS2
SCHEMBL12308318 0.87 ESR1 (0.89) ESR1ESR2PTGS2
SCHEMBL7457759 0.84 ESR1 (0.85) ESR1ESR2ENPP1
Hydrochloric Acid SCHEMBL7457698 0.83 ESR1 (0.84) ESR1ESR2ENPP1
SCHEMBL3743164 0.82 ESR1 (1.00) ESR1ESR2PTGS2
Hydrochloric Acid SCHEMBL3807019 0.82 ESR1 (1.00) ESR1ESR2PTGS2
SCHEMBL20442774 0.81 ESR1 (0.66) ESR1ESR2
SCHEMBL7517965 0.81 ESR1 (0.98) ESR1ESR2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170114052-A1 COMPOSITIONS AND METHODS FOR TREATING ESTROGEN-RELATED MEDICAL DISORDERS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2017-04-27 US disclosed
US-20150284357-A1 COMPOSITIONS AND METHODS FOR TREATING ESTROGEN-RELATED MEDICAL DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150284357-A1 COMPOSITIONS AND METHODS FOR TREATING ESTROGEN-RELATED MEDICAL DISORDERS HSD17B11, CYP19A1, ESR1 ESR1 3/4885ESR2 5/4885LTA4H 1393/4885
US-20170114052-A1 COMPOSITIONS AND METHODS FOR TREATING ESTROGEN-RELATED MEDICAL DISORDERS HSD17B11, CYP19A1, ESR1 ESR1 3/4885ESR2 5/4885LTA4H 1393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.