SCHEMBL17159262

SCHEMBL17159262

Cc1sc(Br)cc1C1CC1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 5/20 0.39
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
DAO P14920 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM1A O60341 7/20 0.34
STING1 Q86WV6 2/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 1/20 0.33
GRM2 Q14416 1/20 0.33
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
TBXA2R P21731 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
PTGER1 P34995 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17159263 1.00 FFAR1 (0.39) FFAR1KDM4EMEN1ALDH1A1MAPT
SCHEMBL17159024 0.80 CA1 (0.42) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL17159025 0.80 CA1 (0.42) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL17164904 0.78 KDM1A (0.42) KDM1A
SCHEMBL17164902 0.78 KDM1A (0.42) KDM1A
SCHEMBL26186746 0.72 HTR2A (0.51) FFAR1ALDH1A1KMT2AGRM2
SCHEMBL17159041 0.72 KDM1A (0.30) KDM1A
SCHEMBL17159039 0.72 KDM1A (0.30) KDM1A
SCHEMBL17164839 0.72 KDM1A (0.34) KDM1A
SCHEMBL17158779 0.69 DAO (0.41) FFAR1KDM4EALDH1A1DAOKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240317733-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2024-09-26 US disclosed
US-20210179603-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2021-06-17 US disclosed
US-10968213-B2 Cyclopropanamine compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-04-06 US disclosed
US-20190315735-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2019-10-17 US disclosed
US-10414761-B2 Cyclopropanamine compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2019-09-17 US disclosed
US-10053456-B2 Cyclopropanamine compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-08-21 US disclosed
US-20180162853-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2018-06-14 US disclosed
US-9920047-B2 Cyclopropanamine compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-03-20 US disclosed
US-9718814-B2 Cyclopropanamine compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-01 US disclosed
US-9714241-B2 Cyclopropanamine compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-07-25 US disclosed
EP-3129369-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2017-02-15 EP disclosed
US-20170029417-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-02-02 US disclosed
US-20170001994-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2017-01-05 US disclosed
US-9487511-B2 Cyclopropanamine compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-11-08 US disclosed
US-20160311814-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2016-10-27 US disclosed
US-20160311808-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2016-10-27 US disclosed
WO-2015156417-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-10-15 WO disclosed
US-20150291577-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190315735-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20160311808-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20180162853-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-10053456-B2 Cyclopropanamine compound and use thereof KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20210179603-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20240317733-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1147/4885KDM4E 13/4885MEN1 1729/4885
US-10968213-B2 Cyclopropanamine compound and use thereof KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20170001994-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-10414761-B2 Cyclopropanamine compound and use thereof KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20150291577-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20170029417-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885
US-20160311814-A1 CYCLOPROPANAMINE COMPOUND AND USE THEREOF KDM1A, KDM1B, KDM2A FFAR1 1287/4885KDM4E 14/4885MEN1 1645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.