SCHEMBL17166275

SCHEMBL17166275

O=C(Nc1ccc(Br)cc1C(=O)O)c1ccc(C(=O)Nc2ccc(Br)cc2C(=O)O)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 4/20 0.73
AKR1C1 Q04828 4/20 0.73
AKR1C4 P17516 1/20 0.73
AKR1C3 P42330 1/20 0.73
KCNK2 O95069 2/20 0.72
KCNK10 P57789 2/20 0.72
MAPT P10636 6/20 0.69
TDP1 Q9NUW8 4/20 0.64
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
ABL1 P00519 1/20 0.64
TSHR P16473 1/20 0.64
RIN1 Q13671 1/20 0.64
DHODH Q02127 1/20 0.62
ALDH1A1 P00352 1/20 0.60
HTT P42858 1/20 0.60
KDM4E B2RXH2 1/20 0.57
ACLY P53396 1/20 0.57
PKM P14618 1/20 0.57
GRIK1 P39086 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6348852 0.95 AKR1C2 (0.72) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL9513479 0.93 MAPT (0.80) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL6360570 0.92 KCNK2 (0.68) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL1307201 0.92 KCNK2 (0.64) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL6350407 0.92 KCNK2 (0.64) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL6353351 0.91 SERPINE1 (0.71) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL6357922 0.91 MAPT (0.81) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL17166040 0.91 MEN1 (0.68) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL20512990 0.91 SERPINE1 (0.66) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2
SCHEMBL6353673 0.90 KCNK2 (0.62) AKR1C2AKR1C1AKR1C4AKR1C3KCNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9155792-B2 RecA inhibitors with antibiotic activity, compositions and methods of use TRUSTEES OF BOSTON UNIVERSITY (US) 2015-10-13 US disclosed