SCHEMBL1717767

SCHEMBL1717767

CC[C@H](NC(=O)c1c(CN2CCN(CCN3CCOCC3)CC2)n(-c2cccc(F)c2)c(=O)c2ccccc12)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 6/20 0.45
KCNK3 O14649 12/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
HSD17B10 Q99714 1/20 0.42
RCE1 Q9Y256 1/20 0.42
TACR2 P21452 3/20 0.41
OPRM1 P35372 2/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719009 0.94 TACR3 (0.47) TACR3KCNK3TACR2OPRM1
SCHEMBL1717248 0.93 TACR3 (0.49) TACR3KCNK3TACR2OPRM1
SCHEMBL1717754 0.93 KCNK3 (0.41) TACR3KCNK3TACR2OPRM1
SCHEMBL1717906 0.92 TACR3 (0.46) TACR3KCNK3ALDH1A1GAATACR2
SCHEMBL1717606 0.92 GAA (0.49) TACR3KCNK3KDM4EUSP2ALDH1A1
SCHEMBL1717731 0.92 KCNK3 (0.43) TACR3KCNK3KDM4EALDH1A1GAA
SCHEMBL1717245 0.91 KCNK3 (0.45) TACR3KCNK3TACR2OPRM1
SCHEMBL1717260 0.91 TACR3 (0.45) TACR3KCNK3TACR2OPRM1
SCHEMBL1717510 0.90 TACR3 (0.44) TACR3KCNK3ALDH1A1GAAHSD17B10
SCHEMBL1717745 0.90 TACR3 (0.47) TACR3KCNK3ALDH1A1GAATACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP claimed
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP disclosed