SCHEMBL1718017

SCHEMBL1718017

CC[C@H](NC(=O)c1c(CN2CCN(CCN3CCCCC3)CC2)n(-c2cccc(C)c2)c(=O)c2ccccc12)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 6/20 0.49
TACR2 P21452 5/20 0.49
OPRM1 P35372 4/20 0.45
KCNK3 O14649 12/20 0.42
TRPV4 Q9HBA0 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1717592 0.99 TACR3 (0.48) TACR3TACR2OPRM1KCNK3TRPV4
SCHEMBL1717606 0.93 GAA (0.49) TACR3TACR2OPRM1KCNK3ALDH1A1
SCHEMBL1717394 0.93 TACR3 (0.54) TACR3TACR2OPRM1KCNK3
SCHEMBL1717925 0.92 TACR3 (0.49) TACR3TACR2OPRM1KCNK3TRPV4
SCHEMBL1718258 0.92 TACR3 (0.53) TACR3TACR2OPRM1KCNK3
SCHEMBL1717248 0.91 TACR3 (0.49) TACR3TACR2OPRM1KCNK3TRPV4
SCHEMBL1717467 0.91 TACR3 (0.42) TACR3TACR2OPRM1KCNK3ALDH1A1
SCHEMBL1717938 0.91 TACR3 (0.48) TACR3TACR2OPRM1KCNK3TRPV4
SCHEMBL1719009 0.91 TACR3 (0.47) TACR3TACR2OPRM1KCNK3TRPV4
SCHEMBL1724094 0.90 TACR3 (0.44) TACR3TACR2OPRM1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP claimed
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP disclosed