SCHEMBL1718098

SCHEMBL1718098

CCOC(=O)ON1CCN(Cc2c(C(=O)NC(CC)c3ccccc3)c3ccccc3c(=O)n2-c2ccccc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 16/20 0.43
TACR2 P21452 10/20 0.43
OPRM1 P35372 5/20 0.43
MAPT P10636 2/20 0.40
NPSR1 Q6W5P4 3/20 0.40
TSHR P16473 2/20 0.40
P4HB P07237 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP2D6 P10635 1/20 0.39
TACR1 P25103 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
NFKB1 P19838 1/20 0.39
MAPK1 P28482 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719117 0.93 TACR3 (0.42) TACR3TACR2OPRM1MAPTNPSR1
SCHEMBL1718106 0.90 TACR3 (0.42) TACR3TACR2OPRM1CYP1A2CYP3A4
SCHEMBL1716895 0.89 TACR3 (0.45) TACR3TACR2OPRM1MAPTNPSR1
SCHEMBL1718399 0.88 TACR3 (0.43) TACR3TACR2OPRM1NPSR1TSHR
SCHEMBL1718231 0.87 TACR3 (0.49) TACR3TACR2OPRM1NPSR1TSHR
SCHEMBL1717859 0.86 TACR3 (0.48) TACR3TACR2OPRM1NPSR1TSHR
SCHEMBL1717555 0.86 TACR3 (0.48) TACR3TACR2OPRM1MAPTNPSR1
SCHEMBL1717937 0.86 TACR3 (0.54) TACR3TACR2OPRM1TSHRCYP1A2
SCHEMBL1718057 0.86 TACR3 (0.56) TACR3TACR2OPRM1TSHRCYP1A2
SCHEMBL1717030 0.85 KMT2A (0.51) TACR3TACR2OPRM1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150534-B1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS LUNDBECK & CO AS H (DK) 2012-01-11 EP claimed