SCHEMBL1719573

SCHEMBL1719573

Cc1cc(C(=O)O)ccc1NC(=O)CSc1nnc(Br)n1-c1ccc(C2CC2)c2ccccc12

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 12/20 0.65
CYP2C9 P11712 3/20 0.65
CYP2C19 P33261 3/20 0.65
CYP3A4 P08684 2/20 0.65
CYP2D6 P10635 2/20 0.65
CYP1A2 P05177 1/20 0.65
SLC22A11 Q9NSA0 1/20 0.65
SLC2A9 Q9NRM0 3/20 0.60
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.44
THRB P10828 1/20 0.44
CCR5 P51681 1/20 0.43
RECQL P46063 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
KDM4E B2RXH2 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL253614 0.93 SLC22A12 (0.62) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10029207 0.92 SLC22A12 (0.53) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL248221 0.91 SLC22A12 (0.65) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL29376753 0.91 SLC22A12 (0.65) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
Potassium SCHEMBL30892115 0.90 SLC22A12 (0.64) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL14921536 0.90 SLC22A12 (0.64) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10029331 0.88 SLC22A12 (0.49) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL249261 0.87 SLC22A12 (0.66) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL12056187 0.85 SLC22A12 (0.64) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10029197 0.84 SLC22A12 (0.51) SLC22A12CYP2C9CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1789039-B1 S-TRIAZOLYL ALPHA -MERCAPTOACETANILDES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE ARDEA BIOSCIENCES INC (US) 2012-01-11 EP claimed