SCHEMBL17196804

SCHEMBL17196804

C=CC(=O)Nc1cc(Nc2ncc(Cl)c(NC3CNC3)n2)c(OC)cc1N1CCC(N(C)C)CC1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.72
ALK Q9UM73 1/20 0.60
INSR P06213 1/20 0.59
IGF1R P08069 1/20 0.59
KCNH2 Q12809 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17196832 0.94 EGFR (0.74) EGFRALKINSRIGF1RKCNH2
SCHEMBL17196822 0.90 EGFR (0.69) EGFRALKINSRIGF1RKCNH2
SCHEMBL18657438 0.89 EGFR (0.68) EGFRALKINSRIGF1RKCNH2
SCHEMBL18657457 0.89 EGFR (0.68) EGFRALKINSRIGF1RKCNH2
SCHEMBL17196889 0.89 EGFR (0.67) EGFRINSRIGF1RKCNH2
SCHEMBL17196955 0.89 EGFR (0.67) EGFRINSRIGF1RKCNH2
SCHEMBL18657432 0.88 EGFR (0.78) EGFRINSRIGF1RKCNH2
SCHEMBL17196876 0.88 EGFR (0.67) EGFRINSRIGF1RKCNH2
SCHEMBL18657720 0.86 EGFR (0.76) EGFRINSRIGF1RKCNH2
SCHEMBL17196891 0.86 EGFR (0.64) EGFRALKINSRIGF1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3144292-A1 2,3,4,6-TETRA-SUBSTITUTED BENZENE-1,5-DIAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICINAL USE THEREOF SHANGHAI HAIYAN PHARMACEUTICAL TECHNOLOGY CO., LTD (US) 2017-03-22 EP disclosed
WO-2015158233-A1 2,3,4,6-TETRA-SUBSTITUTED BENZENE-1,5-DIAMINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICINAL USE THEREOF 上海海雁医药科技有限公司 2015-10-22 WO disclosed