SCHEMBL17200115

SCHEMBL17200115

CNCC(Nc1nc(C)nc2c(C(N)=O)cccc12)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 17/20 0.76
AURKA O14965 12/20 0.76
AKT1 P31749 8/20 0.75
AURKB Q96GD4 4/20 0.75
INCENP Q9NQS7 4/20 0.75
CYP2C9 P11712 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10093523 1.00 RPS6KB1 (0.76) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL527690 0.90 RPS6KB1 (0.79) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL527028 0.89 RPS6KB1 (0.73) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL17200096 0.87 RPS6KB1 (0.68) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL10093516 0.87 RPS6KB1 (0.68) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL666292 0.87 RPS6KB1 (1.00) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL14974658 0.86 RPS6KB1 (0.80) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL10093525 0.86 RPS6KB1 (1.00) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL14974401 0.85 RPS6KB1 (0.82) RPS6KB1AURKAAKT1AURKBINCENP
SCHEMBL10093526 0.85 RPS6KB1 (0.82) RPS6KB1AURKAAKT1AURKBINCENP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598492-B1 BICYCLIC AZAHETEROCYCLIC CARBOXAMIDES AS INHIBITORS OF THE KINASE P70S6K MERCK PATENT GMBH (DE) 2015-10-28 EP disclosed