SCHEMBL1720616

SCHEMBL1720616

Cn1nc(CC2CCNCC2)c2c3ccc(F)cc3c(=O)[nH]c21

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.41
PARP1 P09874 5/20 0.39
TNKS O95271 5/20 0.34
TNKS2 Q9H2K2 5/20 0.34
KCNH2 Q12809 3/20 0.34
BRD3 Q15059 2/20 0.33
PLK1 P53350 1/20 0.33
JAK2 O60674 1/20 0.32
BRD4 O60885 1/20 0.32
ATAD2 Q6PL18 1/20 0.32
PLAT P00750 1/20 0.32
SLC6A2 P23975 1/20 0.32
CTSC P53634 1/20 0.32
KDR P35968 1/20 0.32
NMT1 P30419 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1717425 0.99 SLC6A4 (0.41) SLC6A4PARP1TNKSTNKS2KCNH2
SCHEMBL1719934 0.90 PARP1 (0.41) PARP1TNKSTNKS2JAK2NMT1
SCHEMBL1720253 0.82 PARP1 (0.53) PARP1TNKSTNKS2KCNH2JAK2
Hydrochloric Acid SCHEMBL1720668 0.81 PARP1 (0.53) PARP1TNKSTNKS2KCNH2JAK2
SCHEMBL1720066 0.78 PARP1 (0.39) PARP1TNKSTNKS2PLK1
SCHEMBL1719923 0.78 PARP1 (0.42) PARP1TNKSTNKS2KCNH2PLK1
Hydrochloric Acid SCHEMBL4069890 0.77 PARP1 (0.41) PARP1TNKSTNKS2KCNH2PLK1
SCHEMBL1720207 0.76 PARP1 (0.43) PARP1TNKS
SCHEMBL1720211 0.76 PARP1 (0.43) PARP1TNKS
SCHEMBL1719790 0.76 PARP1 (0.43) PARP1TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1566380-B1 ISOQUINOLINE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI TANABE PHARMA CORP (JP) 2012-01-11 EP claimed
US-7501412-B2 Isoquinoline compounds and medicinal use thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-10 US disclosed
US-7501412-B2 Isoquinoline compounds and medicinal use thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-10 US disclosed