SCHEMBL172069

SCHEMBL172069

CC1=C(C#N)[C@@H](c2ccc(C#N)cc2S(C)(=O)=O)N(C(=O)N2CCC(C(=O)O)CC2)C(=O)N1c1cccc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.67
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8011392 0.93 ELANE (0.69) ELANECYP3A4CYP2C9
SCHEMBL7999190 0.92 ELANE (0.63) ELANECYP3A4CYP2C9
SCHEMBL15473106 0.91 ELANE (0.66) ELANECYP3A4CYP2C9
SCHEMBL8017841 0.91 ELANE (0.67) ELANE
SCHEMBL12859219 0.90 ELANE (0.79) ELANE
SCHEMBL8016374 0.90 ELANE (0.65) ELANECYP3A4CYP2C9
SCHEMBL3724940 0.90 ELANE (0.67) ELANECYP3A4CYP2C9
SCHEMBL170067 0.90 ELANE (0.67) ELANECYP3A4CYP2C9
SCHEMBL124799 0.90 ELANE (0.67) ELANECYP3A4CYP2C9
SCHEMBL121430 0.90 ELANE (0.67) ELANECYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234985-B1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF Bayer Pharma AG (DE) 2012-03-07 EP disclosed
WO-2009080199-A1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed