SCHEMBL1721064

SCHEMBL1721064

CCNC(=O)Nc1ccc(-c2nc3c(c(N4CCOC[C@@H]4C)n2)CN(C2CCN(C(C)(C)C)CC2)C3)cc1F

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTOR P42345 20/20 0.62
PIK3CA P42336 3/20 0.60
CYP3A4 P08684 3/20 0.59
KCNH2 Q12809 1/20 0.53
RPTOR Q8N122 7/20 0.51
MLST8 Q9BVC4 7/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16266021 0.92 MTOR (0.64) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL413950 0.92 MTOR (0.64) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL442763 0.92 MTOR (0.64) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL442175 0.91 MTOR (0.62) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL413960 0.91 MTOR (0.62) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL443656 0.91 MTOR (0.64) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL443657 0.91 MTOR (0.64) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL16109384 0.90 MTOR (0.64) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL16109386 0.90 MTOR (0.64) MTORPIK3CACYP3A4KCNH2RPTOR
SCHEMBL16266037 0.88 MTOR (0.59) MTORPIK3CACYP3A4KCNH2RPTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406258-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS Cellzome Limited (GB) 2012-01-18 EP disclosed
WO-2010103094-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS CELLZOME LIMITED (GB) 2010-09-16 WO disclosed