SCHEMBL17212957

SCHEMBL17212957

Cc1c(O)ccc2c(O)ccnc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.45
CCR5 P51681 3/20 0.45
CCR8 P51685 3/20 0.45
HTT P42858 3/20 0.44
SLC6A2 P23975 1/20 0.44
L3MBTL1 Q9Y468 5/20 0.39
HSP90AA1 P07900 3/20 0.39
NPC1 O15118 2/20 0.39
LMNA P02545 5/20 0.39
KMT2A Q03164 4/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
COMT P21964 1/20 0.38
OPRK1 P41145 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
PKM P14618 1/20 0.37
KDM4E B2RXH2 4/20 0.36
MPI P34949 1/20 0.36
BRD4 O60885 1/20 0.36
METAP2 P50579 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8602817 0.86 CCR1 (0.48) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL16742815 0.82 HSP90AA1 (0.44) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL15010895 0.82 CCR1 (0.41) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL17212936 0.82 KDM4E (0.53) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL1073354 0.82 CCR1 (0.50) CCR1CCR5CCR8HTTSLC6A2
Hydrochloric Acid SCHEMBL11825124 0.80 CCR1 (0.48) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL995835 0.80 MEN1 (0.40) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL15483503 0.80 KDM4E (0.49) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL13328096 0.79 CCR1 (0.75) CCR1CCR5CCR8HTTSLC6A2
SCHEMBL28192061 0.77 TOP2A (0.54) HTTSLC6A2COMTTLR8TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2937339-A1 Macrocylic inhibitors of hepatitis c virus Janssen Sciences Ireland UC (IE) 2015-10-28 EP disclosed