SCHEMBL17220193

SCHEMBL17220193

CN(c1ccccc1)c1nc(N)nc(-c2noc(-c3ccc(COS(C)(=O)=O)nc3)n2)n1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 5/20 0.33
CA9 Q16790 5/20 0.33
ATM Q13315 2/20 0.33
ATR Q13535 2/20 0.33
PRKDC P78527 1/20 0.33
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
S1PR1 P21453 2/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
HDAC1 Q13547 4/20 0.32
HDAC6 Q9UBN7 4/20 0.32
HDAC5 Q9UQL6 4/20 0.32
HDAC8 Q9BY41 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL795256 0.87 ALOX5AP (0.33) CA2CA9ATMATRPRKDC
SCHEMBL10287193 0.84 S1PR1 (0.33) S1PR1BCHEACHEHDAC1HDAC6
SCHEMBL795739 0.84 S1PR1 (0.44) ATRS1PR1BCHEACHEKDM4E
SCHEMBL796180 0.84 ALOX5AP (0.34) S1PR1BCHEACHEHDAC1HDAC6
SCHEMBL795506 0.83 HDAC6 (0.38) S1PR1HDAC1HDAC6HDAC5HDAC8
SCHEMBL795736 0.83 CNR2 (0.35) S1PR1BCHEACHEHDAC1HDAC6
SCHEMBL796335 0.82 ATM (0.33) CA2CA9ATMATRPRKDC
SCHEMBL15477342 0.82 HDAC6 (0.35) S1PR1HDAC1HDAC6HDAC5HDAC8
SCHEMBL797145 0.81 TP53 (0.36) S1PR1BCHEACHEKDM4ENPC1
SCHEMBL10286922 0.80 S1PR1 (0.33) S1PR1BCHEACHEHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616465-B1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2015-11-04 EP disclosed