SCHEMBL172210

SCHEMBL172210

C[C@@H]1CN(C2=Nc3cc(Cl)ccc3Oc3ccccc32)CCN1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 10/20 0.65
DRD4 P21917 6/20 0.65
DRD2 P14416 4/20 0.65
HTR2A P28223 6/20 0.62
ADRA2A P08913 5/20 0.62
HTR1A P08908 5/20 0.62
HRH2 P25021 3/20 0.62
HRH1 P35367 3/20 0.62
CHRM2 P08172 3/20 0.62
CHRM4 P08173 3/20 0.62
CHRM5 P08912 3/20 0.62
CHRM1 P11229 3/20 0.62
CHRM3 P20309 3/20 0.62
DRD1 P21728 3/20 0.62
KCNH2 Q12809 3/20 0.62
HTR2C P28335 3/20 0.62
CYP1A2 P05177 3/20 0.62
CYP3A4 P08684 3/20 0.62
CYP2D6 P10635 3/20 0.62
ADRB2 P07550 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8930455 0.88 HRH4 (0.66) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL2738976 0.84 DRD4 (0.82) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL10125507 0.83 HRH4 (0.62) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL121787 0.83 HRH4 (0.65) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL10125487 0.83 HRH4 (0.60) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL123140 0.83 HRH4 (0.65) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL10125483 0.83 HRH4 (0.62) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL123038 0.83 HRH4 (0.65) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL10125471 0.83 HRH4 (0.60) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL121788 0.83 HRH4 (0.65) HRH4DRD4DRD2HTR2AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137180-B1 DIBENZO [B,F][1,4] OXAZAPINE COMPOUNDS ARYX THERAPEUTICS INC (US) 2012-03-07 EP disclosed