SCHEMBL1722111

SCHEMBL1722111

CC(I)NC(=O)Nc1ccc(-c2nc3c(c(N4CCOCC4C)n2)CNC3)cc1F

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MTOR P42345 20/20 0.46
KCNH2 Q12809 1/20 0.46
PIK3CA P42336 3/20 0.44
CYP3A4 P08684 3/20 0.43
RPTOR Q8N122 2/20 0.41
MLST8 Q9BVC4 2/20 0.41
PIK3R1 P27986 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL411910 0.88 MTOR (0.58) MTORKCNH2PIK3CACYP3A4RPTOR
SCHEMBL442183 0.88 MTOR (0.58) MTORKCNH2PIK3CACYP3A4RPTOR
SCHEMBL1721199 0.88 MTOR (0.58) MTORKCNH2PIK3CACYP3A4RPTOR
Hydrochloric Acid SCHEMBL443870 0.87 MTOR (0.57) MTORKCNH2PIK3CACYP3A4RPTOR
Hydrochloric Acid SCHEMBL443871 0.87 MTOR (0.57) MTORKCNH2PIK3CACYP3A4RPTOR
SCHEMBL1831772 0.81 MTOR (0.60) MTORKCNH2PIK3CACYP3A4RPTOR
SCHEMBL1834821 0.81 MTOR (0.58) MTORKCNH2PIK3CACYP3A4RPTOR
Hydrochloric Acid SCHEMBL3235341 0.80 MTOR (0.57) MTORKCNH2PIK3CACYP3A4RPTOR
SCHEMBL1834135 0.77 MTOR (0.61) MTORKCNH2PIK3CACYP3A4RPTOR
SCHEMBL442034 0.77 MTOR (0.61) MTORKCNH2PIK3CACYP3A4RPTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406258-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS Cellzome Limited (GB) 2012-01-18 EP disclosed
WO-2010103094-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS CELLZOME LIMITED (GB) 2010-09-16 WO disclosed