SCHEMBL172233

SCHEMBL172233

Cc1c(CN2CCN(c3nccnc3N3CCC(CN)CC3)CC2)cnn1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 3/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
SMO Q99835 2/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
CXCR4 P61073 1/20 0.37
GSK3B P49841 1/20 0.36
ALPI P09923 1/20 0.36
ALPG P10696 1/20 0.36
CHEK1 O14757 2/20 0.36
CHEK2 O96017 2/20 0.36
ALDH1A1 P00352 1/20 0.36
RET P07949 1/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
TRPC5 Q9UL62 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL122179 0.89 PDE10A (0.43) CNR1CNR2SMODRD2DRD4
Hydrochloric Acid SCHEMBL125616 0.88 PDE10A (0.43) CNR1CNR2SMODRD2DRD4
SCHEMBL172372 0.87 CNR1 (0.42) CNR1CNR2SMODRD2DRD4
SCHEMBL170286 0.87 CNR1 (0.42) CNR1CNR2SMODRD2DRD4
SCHEMBL170321 0.87 CNR1 (0.40) CNR1CNR2SMODRD2DRD4
SCHEMBL12742533 0.87 CNR1 (0.40) CNR1CNR2SMODRD2DRD4
Hydrochloric Acid SCHEMBL123007 0.86 CNR1 (0.42) CNR1CNR2SMODRD2DRD4
SCHEMBL172325 0.86 CNR1 (0.42) CNR1CNR2SMODRD2DRD4
Hydrochloric Acid SCHEMBL124394 0.86 CNR1 (0.42) CNR1CNR2SMODRD2DRD4
Hydrochloric Acid SCHEMBL123983 0.86 CNR1 (0.39) CNR1CNR2SMODRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2201002-B1 5-HT7 RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2012-03-07 EP disclosed
WO-2009048765-A1 5-HT7 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2009-04-16 WO disclosed