SCHEMBL17226871

SCHEMBL17226871

Fc1ccc(-c2cnc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)cn1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 17/20 0.81
CYP3A4 P08684 3/20 0.75
LRRK2 Q5S007 3/20 0.75
CYP2D6 P10635 2/20 0.75
CYP2C9 P11712 1/20 0.75
DYRK1A Q13627 3/20 0.73
DYRK2 Q92630 2/20 0.73
DYRK1B Q9Y463 2/20 0.73
CLK1 P49759 1/20 0.69
SGK1 O00141 1/20 0.58
IKBKB O14920 1/20 0.58
AURKA O14965 1/20 0.58
CHUK O15111 1/20 0.58
PRKAB2 O43741 1/20 0.58
ROCK2 O75116 1/20 0.58
ABL1 P00519 1/20 0.58
NTRK1 P04629 1/20 0.58
INSR P06213 1/20 0.58
LCK P06239 1/20 0.58
CDK1 P06493 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL723789 0.90 MAP3K11 (1.00) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL723923 0.86 MAP3K11 (1.00) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL721629 0.85 MAP3K11 (1.00) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL722261 0.85 MAP3K11 (0.80) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL720976 0.84 MAP3K11 (1.00) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL12763475 0.84 MAP3K11 (0.83) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL724304 0.84 MAP3K11 (0.83) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL721195 0.83 MAP3K11 (1.00) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL721794 0.83 MAP3K11 (1.00) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9
SCHEMBL3767742 0.81 MAP3K11 (0.78) MAP3K11CYP3A4LRRK2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3037421-A1 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2016-06-29 EP disclosed
EP-2379561-B1 MLK INHIBITORS AND METHODS OF USE UNIV ROCHESTER (US) 2015-11-04 EP disclosed