SCHEMBL17236509

SCHEMBL17236509

NC(=O)c1ccnc2[nH]c(-c3ccc(-c4ccc(CC5CC5)cc4)cc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.47
PARP1 P09874 19/20 0.46
PARP2 Q9UGN5 6/20 0.44
DHODH Q02127 4/20 0.43
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17236507 0.90 DHODH (0.43) CHEK2PARP1DHODH
SCHEMBL17224985 0.81 PARP1 (0.64) CHEK2PARP1PARP2DHODH
SCHEMBL17224854 0.79 PARP1 (0.49) PARP1PARP2DHODH
SCHEMBL13778349 0.78 PARP1 (0.52) CHEK2PARP1PARP2DHODH
SCHEMBL17224941 0.75 PARP1 (0.60) CHEK2PARP1DHODHHDAC3HDAC4
SCHEMBL4970975 0.74 PARP1 (0.72) PARP1PARP2DHODH
SCHEMBL17224889 0.71 DHODH (0.62) PARP1DHODH
SCHEMBL4975139 0.70 PARP1 (0.75) PARP1PARP2
SCHEMBL3150584 0.70 PARP1 (0.71) CHEK2PARP1PARP2DHODH
SCHEMBL17224960 0.69 DHODH (0.57) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015166398-A1 3H-IMIDAZO[4,5-B]PYRIDINE DERIVATIVES AS DIHYDROOROTATE DEHYDROGENASE INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-11-05 WO disclosed