SCHEMBL172519

SCHEMBL172519

CCCC(N)c1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.41
TDO2 P48775 2/20 0.41
CFD P00746 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
GNRHR P30968 1/20 0.38
BCDIN3D Q7Z5W3 3/20 0.36
MC4R P32245 3/20 0.36
PSIP1 O75475 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728815 0.89 IDO1 (0.39) IDO1TDO2CFDGNRHRBCDIN3D
SCHEMBL1727508 0.89 IDO1 (0.39) IDO1TDO2CFDGNRHRBCDIN3D
SCHEMBL4672694 0.85 IDO1 (0.44) IDO1TDO2CFDGNRHRBCDIN3D
SCHEMBL3680376 0.85 AOC3 (0.38) CFD
SCHEMBL30682632 0.83 IDO1 (0.40) IDO1TDO2MC4RPSIP1CYP3A4
SCHEMBL30682733 0.83 IDO1 (0.40) IDO1TDO2MC4RPSIP1CYP3A4
SCHEMBL5205809 0.83 IDO1 (0.40) IDO1TDO2MC4RPSIP1CYP3A4
SCHEMBL1728822 0.83 IDO1 (0.40) IDO1TDO2MC4RPSIP1CYP3A4
SCHEMBL1727474 0.83 IDO1 (0.40) IDO1TDO2MC4RPSIP1CYP3A4
SCHEMBL30682588 0.83 IDO1 (0.40) IDO1TDO2MC4RPSIP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255738-B1 GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO NEUROCRINE BIOSCIENCES INC (US) 2012-03-07 EP disclosed