SCHEMBL17255671

SCHEMBL17255671

NC(=O)c1cccc2[nH]c(-c3cccc(C(F)(F)F)c3C(=O)NC3CCCCC3)nc12

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.64
PARP2 Q9UGN5 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.50
PTGES O14684 1/20 0.48
MAP4K4 O95819 1/20 0.48
CSF1R P07333 1/20 0.48
PIM1 P11309 1/20 0.48
CLK2 P49760 1/20 0.48
MAP4K2 Q12851 1/20 0.48
DYRK1A Q13627 1/20 0.48
MINK1 Q8N4C8 1/20 0.48
AURKB Q96GD4 1/20 0.48
MAP4K5 Q9Y4K4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7320347 0.79 PARP1 (1.00) PARP1PARP2MAP4K4PIM1CLK2
SCHEMBL12662024 0.77 PARP1 (0.62) PARP1PARP2SMN1; SMN2PTGES
SCHEMBL12662011 0.77 PARP1 (0.61) PARP1PARP2SMN1; SMN2PTGES
SCHEMBL12673317 0.72 PARP1 (0.66) PARP1SMN1; SMN2PTGES
SCHEMBL3150588 0.71 PARP1 (0.61) PARP1PARP2MAP4K4CSF1RPIM1
SCHEMBL12662055 0.71 PARP1 (0.51) PARP1PARP2SMN1; SMN2PTGESMAP4K4
SCHEMBL12662033 0.71 PARP1 (0.51) PARP1PARP2SMN1; SMN2PTGESMAP4K4
SCHEMBL12662054 0.71 PARP1 (0.51) PARP1PARP2SMN1; SMN2PTGESMAP4K4
SCHEMBL25217212 0.70 PKN1 (0.66) PARP1PARP2SMN1; SMN2MAP4K4PIM1
SCHEMBL30440661 0.70 PKN1 (0.66) PARP1PARP2SMN1; SMN2MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2746265-B1 HETEROCYCLIC DERIVATIVE AS MICROSOMAL PROSTAGLANDIN E SYNTHASE (mPGEs) INHIBITOR NIPPON SHINYAKU CO LTD (JP) 2015-11-18 EP claimed