SCHEMBL1725644

SCHEMBL1725644

Cn1cc(-c2cccc(-n3ncc4cccc(F)c4c3=O)c2CO)cc(NC2=NCCCO2)c1=O

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.54
KCNH2 Q12809 2/20 0.44
YES1 P07947 1/20 0.43
FGR P09769 1/20 0.43
TEC P42680 1/20 0.43
BMX P51813 1/20 0.43
SLK Q9H2G2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1726667 0.91 BTK (0.67) BTKKCNH2
SCHEMBL3051457 0.86 BTK (0.68) BTKKCNH2
SCHEMBL1725882 0.79 BTK (0.65) BTKKCNH2
SCHEMBL1727066 0.79 BTK (0.65) BTKKCNH2
SCHEMBL13178759 0.78 BTK (0.52) BTKKCNH2YES1FGRTEC
SCHEMBL18199004 0.78 BTK (0.70) BTKKCNH2
SCHEMBL1725805 0.75 BTK (0.55) BTK
SCHEMBL18198976 0.73 BTK (0.67) BTKKCNH2
SCHEMBL3052177 0.73 BTK (0.71) BTKKCNH2
SCHEMBL1729634 0.72 BTK (0.72) BTKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403846-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE F. Hoffmann-La Roche AG (CH) 2012-01-11 EP disclosed