SCHEMBL1727587

SCHEMBL1727587

CN1Cc2nc(-c3ccc(NC(=O)Oc4ccccc4)cc3)nc(N3CCOCC3S(C)(=O)=O)c2C1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTOR P42345 20/20 0.49
PIK3CA P42336 3/20 0.45
CYP3A4 P08684 2/20 0.44
RPTOR Q8N122 1/20 0.43
MLST8 Q9BVC4 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1727589 1.00 MTOR (0.49) MTORPIK3CACYP3A4RPTORMLST8
SCHEMBL442051 0.89 MTOR (0.56) MTORPIK3CACYP3A4RPTORMLST8
SCHEMBL411892 0.89 MTOR (0.56) MTORPIK3CACYP3A4RPTORMLST8
SCHEMBL412933 0.74 MTOR (0.62) MTORPIK3CACYP3A4RPTORMLST8
SCHEMBL442113 0.74 MTOR (0.62) MTORPIK3CACYP3A4RPTORMLST8
SCHEMBL13257089 0.73 PIK3CA (0.72) MTORPIK3CA
SCHEMBL413813 0.72 MTOR (0.64) MTORPIK3CACYP3A4RPTORMLST8
SCHEMBL443639 0.72 MTOR (0.64) MTORPIK3CACYP3A4RPTORMLST8
SCHEMBL3591943 0.72 PIK3CA (0.72) MTORPIK3CA
SCHEMBL411879 0.72 MTOR (0.79) MTORPIK3CACYP3A4RPTORMLST8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406258-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS Cellzome Limited (GB) 2012-01-18 EP disclosed
WO-2010103094-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS CELLZOME LIMITED (GB) 2010-09-16 WO disclosed