SCHEMBL17277136

SCHEMBL17277136

CN(N)CCCOc1cccc(-c2cc3cn(-c4ccc(CNC(=O)CCNC(=N)N)cc4)c(=O)nc3[nH]2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.34
CHUK O15111 4/20 0.34
IKBKB O14920 2/20 0.34
F7 P08709 3/20 0.33
ALDH1A1 P00352 1/20 0.33
KIT P10721 4/20 0.33
SUCNR1 Q9BXA5 1/20 0.33
F3 P13726 2/20 0.32
F2 P00734 1/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
ROCK2 O75116 1/20 0.32
CYP2D6 P10635 1/20 0.32
ROCK1 Q13464 1/20 0.32
DYRK3 O43781 1/20 0.32
MAP4K4 O95819 1/20 0.32
PIM1 P11309 1/20 0.32
RPS6KB1 P23443 1/20 0.32
CSNK2A1 P68400 1/20 0.32
PKN2 Q16513 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565 0.95 CHEK2 (0.39) CHEK2CHUKIKBKBF7ALDH1A1
SCHEMBL14357 0.91 KIT (0.35) CHUKIKBKBF7KITSUCNR1
SCHEMBL14216 0.85 CHEK2 (0.39) CHEK2CHUKF7F3CYP3A4
SCHEMBL12062173 0.82 KCNA5 (0.35) CHEK2CHUKKITINSRMAPK8
SCHEMBL17277137 0.82 TLR7 (0.36) KDM4EABL1EGFRSRCABL2
SCHEMBL14300 0.82 EGFR (0.34) KITKDM4EABL1EGFRSRC
SCHEMBL12062128 0.82 SRC (0.38) CHUKKITINSRMAPK8CAMKK2
SCHEMBL14477 0.81 SRC (0.35) ALDH1A1KITKDM4EABL1EGFR
SCHEMBL13966 0.81 SRC (0.38) CHUKKITINSRMAPK8CAMKK2
SCHEMBL20082539 0.80 SRC (0.34) KITKDM4EABL1EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9193731-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2015-11-24 US disclosed