SCHEMBL17277682

SCHEMBL17277682

CC(C)(C)OC(=O)N1CCCCC1c1nc2ccc(Br)cc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.55
HCRTR2 O43614 19/20 0.55
CHEK2 O96017 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12327656 1.00 HCRTR1 (0.55) HCRTR1HCRTR2CHEK2
SCHEMBL16215441 1.00 HCRTR1 (0.55) HCRTR1HCRTR2CHEK2
SCHEMBL1293520 0.97 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL38658108 0.97 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL204028 0.97 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL2706134 0.97 HCRTR1 (0.58) HCRTR1HCRTR2
SCHEMBL12567373 0.92 HCRTR1 (0.47) HCRTR1HCRTR2CHEK2
SCHEMBL1357197 0.89 HCRTR1 (0.56) HCRTR1HCRTR2CHEK2
SCHEMBL1357196 0.89 HCRTR1 (0.56) HCRTR1HCRTR2CHEK2
SCHEMBL1982286 0.89 HCRTR1 (0.49) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545060-B1 FUSED TRICYCLIC SILYL COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME (US) 2015-11-25 EP disclosed