Epicorticosterone

Epicorticosterone

SCHEMBL17287012

C[C@]12CCC(=O)C=C1CC[C@@H]1C2[C@@H](O)C[C@@]2(C)C1CC[C@@H]2C(=O)CO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 1.00
HIF1A Q16665 6/20 1.00
NR3C2 P08235 6/20 1.00
LMNA P02545 4/20 1.00
SHBG P04278 4/20 1.00
SERPINA6 P08185 4/20 1.00
HSD17B10 Q99714 4/20 1.00
CYP3A4 P08684 4/20 1.00
MAPT P10636 3/20 1.00
MAPK1 P28482 2/20 1.00
NFKB1 P19838 2/20 1.00
BLM P54132 1/20 1.00
CYP2C9 P11712 1/20 1.00
TSHR P16473 1/20 1.00
SLC22A2 O15244 1/20 1.00
SLC22A1 O15245 1/20 1.00
SLC22A3 O75751 1/20 1.00
THPO P40225 1/20 1.00
MTOR P42345 1/20 1.00
SIGMAR1 Q99720 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Epicorticosterone SCHEMBL19465689 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Corticosterone SCHEMBL22612 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Epicorticosterone SCHEMBL14592717 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Corticosterone SCHEMBL5669349 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Epicorticosterone SCHEMBL4380327 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Epicorticosterone SCHEMBL20058459 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Epicorticosterone SCHEMBL9070639 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Epicorticosterone SCHEMBL15920519 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Epicorticosterone SCHEMBL21168995 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG
Epicorticosterone SCHEMBL20242898 1.00 SMN1; SMN2 (1.00) SMN1; SMN2HIF1ANR3C2LMNASHBG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023183807-A1 AQUEOUS PHARMACEUTICAL FORMULATION OF HYDROCORTISONE SODIUM PHOSPHATE AND MONOTHIOGLYCEROL ANTARES PHARMA, INC. (US) 2023-09-28 WO disclosed
US-10813939-B2 Bromodomain inhibitor as adjuvant in cancer immunotherapy H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2020-10-27 US disclosed
US-10676484-B2 Compositions and methods for treating leukemia DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-06-09 US disclosed
US-10407441-B2 Compositions and methods for treating neoplasia, inflammatory disease and other disorders DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-09-10 US disclosed
US-20180222917-A1 COMPOSITIONS AND METHODS FOR TREATING LEUKEMIA COLD SPRING HARBOR LABORATORY 2018-08-09 US disclosed
US-20170360801-A1 BROMODOMAIN INHIBITOR AS ADJUVANT IN CANCER IMMUNOTHERAPY H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. 2017-12-21 US disclosed
US-9763956-B2 Diagnostic and treatment methods in subjects having or at risk of developing resistance to cancer therapy THE BROAD INSTITUTE, INC. (US) 2017-09-19 US disclosed
US-9757385-B2 Method of treating leukemia using pharmaceutical formulation containing thienotriazolodiazepine compounds MERCK SHARP & DOHME CORP. (US) 2017-09-12 US disclosed
US-20170157141-A1 METHOD OF TREATING LEUKEMIA USING PHARMACEUTICAL FORMULATION CONTAINING THIENOTRIAZOLODIAZEPINE COMPOUNDS ONCOETHIX GMBH (CH) 2017-06-08 US disclosed
US-20170145013-A1 DIHYDROPTERIDINONE DERIVATIVES AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2017-05-25 US disclosed
US-20170029437-A1 Compositions and Methods for Treating Neoplasia, Inflammatory Disease and Other Disorders NATIONAL INSTITUTES OF HEALTH- DIRECTOR DEITR 2017-02-02 US disclosed
US-20150335704-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING GELS AND METHODS FOR FABRICATING THEREOF IMPRIMIS PHARMACEUTICALS, INC. (US) 2015-11-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170157141-A1 METHOD OF TREATING LEUKEMIA USING PHARMACEUTICAL FORMULATION CONTAINING THIENOTRIAZOLODIAZEPINE COMPOUNDS CCR10, HRH4, H1-10 SMN1; SMN2 1191/4885HIF1A 2998/4885NR3C2 147/4885
US-10813939-B2 Bromodomain inhibitor as adjuvant in cancer immunotherapy BRDT, BRD4, BRD1 SMN1; SMN2 4177/4885HIF1A 2842/4885NR3C2 3266/4885
US-10407441-B2 Compositions and methods for treating neoplasia, inflammatory disease and other disorders BRPF3, EP300, BRD3 SMN1; SMN2 4030/4885HIF1A 1270/4885NR3C2 689/4885
US-10676484-B2 Compositions and methods for treating leukemia MCL1, ABL1, FLT3 SMN1; SMN2 2078/4885HIF1A 221/4885NR3C2 3040/4885
US-20170360801-A1 BROMODOMAIN INHIBITOR AS ADJUVANT IN CANCER IMMUNOTHERAPY BRDT, BRD4, BRD1 SMN1; SMN2 4177/4885HIF1A 2842/4885NR3C2 3266/4885
US-20180222917-A1 COMPOSITIONS AND METHODS FOR TREATING LEUKEMIA MCL1, ABL1, FLT3 SMN1; SMN2 2078/4885HIF1A 221/4885NR3C2 3040/4885
US-20170145013-A1 DIHYDROPTERIDINONE DERIVATIVES AND USES THEREOF BRDT, BRD4, BRD3 SMN1; SMN2 4517/4885HIF1A 2068/4885NR3C2 288/4885
US-20170029437-A1 Compositions and Methods for Treating Neoplasia, Inflammatory Disease and Other Disorders BRPF3, EP300, BRD3 SMN1; SMN2 4030/4885HIF1A 1270/4885NR3C2 689/4885
US-20150335704-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING GELS AND METHODS FOR FABRICATING THEREOF PDE6G, PDE6D, PDE6H SMN1; SMN2 2700/4885HIF1A 3072/4885NR3C2 4692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.