SCHEMBL17295201

SCHEMBL17295201

Cc1cc(NCc2cncn2C)ccc1C#N

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAP3K8 P41279 3/20 0.49
IDH1 O75874 2/20 0.43
BRD4 O60885 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.36
PRKDC P78527 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572173 0.85 FNTA (0.50)
SCHEMBL15134221 0.80 MAP3K8 (0.46) MAP3K8
SCHEMBL7572286 0.78 FNTA (0.57)
SCHEMBL28748316 0.71 HTT (0.46) IDH1ABCG2PRKDC
SCHEMBL17295517 0.68 IDH1 (0.43) MAP3K8IDH1
SCHEMBL20714811 0.67 HTT (0.50) IDH1ABCG2
SCHEMBL26989819 0.67 IDH1 (0.40) IDH1ABCG2PRKDC
SCHEMBL46652 0.67
SCHEMBL12117937 0.65 ABCG2 (0.46) IDH1ABCG2PRKDC
SCHEMBL24896332 0.65 HTT (0.47) IDH1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015181272-A1 RAB GERANYLGERANYL TRANSFERASE INHIBITORS LEAD DISCOVERY CENTER GMBH (DE) 2015-12-03 WO disclosed
WO-2015181272-A1 RAB GERANYLGERANYL TRANSFERASE INHIBITORS LEAD DISCOVERY CENTER GMBH (DE) 2015-12-03 WO disclosed