SCHEMBL1730211

SCHEMBL1730211

CCOc1cc2c(nc1C(=O)NC)C(=N)N(CC(=O)c1cc(-c3ccncc3)c(OC)c(C(C)(C)C)c1)C2

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2R P25116 15/20 0.45
CYP1A1 P04798 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP1B1 Q16678 2/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL5481445 0.99 F2R (0.46) F2RCYP1A1CYP1A2CYP2D6CYP1B1
Bromide SCHEMBL1730631 0.88 F2R (0.52) F2RKDM4ENPC1MAPTRAB9A
Bromide SCHEMBL1732302 0.87 F2R (0.45) F2RKDM4ENPC1MAPTRAB9A
Bromide SCHEMBL1732111 0.86 F2R (0.46) F2R
SCHEMBL1729743 0.86 F2R (0.48) F2RMAPTCYP3A4
SCHEMBL14449121 0.85 F2R (0.49) F2RCYP3A4
Trifluoroacetic Acid SCHEMBL1729328 0.85 F2R (0.51) F2RMAPT
Bromide SCHEMBL1732795 0.85 F2R (0.47) F2RKDM4ENPC1MAPTRAB9A
Bromide SCHEMBL1732515 0.85 F2R (0.49) F2RKDM4ENPC1MAPTRAB9A
Hydrochloric Acid SCHEMBL1730634 0.85 F2R (0.49) F2RCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8951502-B2 Method of dynamic nuclear polarisation (DNP) GE HEALTHCARE AS (NO) 2015-02-10 US disclosed
EP-1954321-B1 METHOD OF DYNAMIC NUCLEAR POLARISATION (DNP) USING A TRITYL RADICAL AND A PARAMAGNETIC METAL ION GE HEALTHCARE AS (NO) 2011-11-23 EP disclosed
EP-1391451-B1 2-IMINOPYRROLIDINE DERIVATES EISAI R&D MAN CO LTD (JP) 2011-11-23 EP disclosed
EP-1954321-A2 METHOD OF DYNAMIC NUCLEAR POLARISATION (DNP) USING A TRITYL RADICAL AND A PARAMAGNETIC METAL ION GE Healthcare AS (NO) 2008-08-13 EP disclosed
WO-2007064226-A2 METHOD OF DYNAMIC NUCLEAR POLARISATION (DNP) USING A TRITYL RADICAL AND A PARAMAGNETIC METAL ION GE HEALTHCARE AS (NO) 2007-06-07 WO disclosed