SCHEMBL1734047

SCHEMBL1734047

C#CC(c1ccc(-c2nc3cc(C#N)cc(C(C)C)c3o2)cc1)C1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CETP P11597 19/20 0.47
KCNH2 Q12809 2/20 0.46
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1735068 0.79 CETP (0.50) CETPKCNH2
SCHEMBL1734851 0.78 CETP (0.51) CETPKCNH2
SCHEMBL3787793 0.77 CETP (0.57) CETPKCNH2
SCHEMBL13082829 0.75 CETP (0.56) CETPKCNH2
SCHEMBL1735063 0.75 ESR1 (0.54) CETPKCNH2ESR1ESR2
SCHEMBL1735106 0.75 CETP (0.54) CETPKCNH2ESR1ESR2
SCHEMBL3690878 0.75 CETP (0.76) CETPKCNH2
SCHEMBL1736290 0.75 ESR1 (0.51) CETPKCNH2ESR1ESR2
SCHEMBL1734951 0.75 CETP (0.52) CETPKCNH2ESR1ESR2
SCHEMBL1734615 0.75 CETP (0.51) CETPKCNH2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954287-B2 CETP INHIBITORS MERCK SHARP & DOHME (US) 2016-02-24 EP disclosed
EP-1954287-B1 CETP INHIBITORS MERCK SHARP & DOHME (US) 2011-11-16 EP disclosed
US-20110262658-A1 PROCESS AND DEVICE FOR TREATING THE COATING OF THERMOPLASTIC RESIN CONTAINERS ZOPPAS MATTEO 2011-10-27 US disclosed