SCHEMBL17340643

SCHEMBL17340643

C=C(NC)c1c(-c2ccc(F)cc2)oc2ccc(-c3cccc(C(=O)NC(C)(C)c4ccc(OC)cc4)c3)cc12

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 4/20 0.44
RCE1 Q9Y256 1/20 0.42
CNR2 P34972 4/20 0.41
BCHE P06276 2/20 0.41
CNR1 P21554 2/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
ATM Q13315 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C8 P10632 2/20 0.39
MAPK1 P28482 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10242009 0.93 ANO1 (0.46) ANO1RCE1CNR2BCHECNR1
SCHEMBL1919008 0.86 CYP3A4 (0.50) CYP3A4CYP2C8KCNH2
SCHEMBL17340642 0.83 CYP3A4 (0.42) ANO1CYP3A4CYP2C8KCNH2
SCHEMBL1919204 0.83 CYP3A4 (0.53) CYP3A4CYP2C8KCNH2
SCHEMBL1918773 0.83 CYP3A4 (0.47) CYP3A4CYP2C8KCNH2
SCHEMBL1918978 0.81 CYP2C8 (0.53) CYP3A4CYP2C8KCNH2
SCHEMBL10241927 0.79 CYP3A4 (0.50) ANO1RCE1CNR2BCHECNR1
SCHEMBL1919864 0.78 CYP3A4 (0.52) CYP3A4CYP2C8KCNH2
SCHEMBL10241997 0.78 CYP3A4 (0.49) ANO1CYP3A4CYP2C8KCNH2
SCHEMBL10242011 0.78 CYP2C8 (0.49) CYP3A4CYP2C8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326633-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2015-12-16 EP disclosed