SCHEMBL1734508

SCHEMBL1734508

NC(=O)c1cc(-c2ccccc2)nc(NCCCCCc2ccccc2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
ASPH Q12797 1/20 0.44
RIOX2 Q8IUF8 1/20 0.44
KDM8 Q8N371 1/20 0.44
EGLN1 Q9GZT9 1/20 0.44
FAAH O00519 2/20 0.43
HRH1 P35367 1/20 0.43
HRH4 Q9H3N8 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
HSD17B10 Q99714 1/20 0.43
DAGLA Q9Y4D2 1/20 0.43
PIK3CB P42338 1/20 0.43
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
CFTR P13569 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1735729 0.95 KDM4E (0.48) KDM4EASPHRIOX2KDM8FAAH
SCHEMBL1734521 0.90 HRH1 (0.52) KDM4EHRH1HRH4ALDH1A1GAA
SCHEMBL1733560 0.87 KDM4E (0.53) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL1734267 0.84 PIK3CB (0.57) KDM4EHRH1HRH4ALDH1A1GAA
SCHEMBL1734127 0.82 KDM4E (0.57) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL1735703 0.81 KDM4E (0.49) KDM4EHRH4ALDH1A1GAAHPGD
SCHEMBL1734332 0.79 KDM4E (0.60) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL1734473 0.79 KDM4E (0.48) KDM4EALDH1A1GAAHPGDTSHR
SCHEMBL1734504 0.79 KDM4E (0.51) KDM4EHRH4ALDH1A1GAAHPGD
SCHEMBL1734154 0.79 IDH1 (0.54) KDM4EALDH1A1GAAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed