SCHEMBL17350161

SCHEMBL17350161

OCC(CO)NCCc1ccc2c(c1)CCc1c-2noc1-c1noc(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.69
S1PR3 Q99500 15/20 0.66
CYP3A4 P08684 1/20 0.53
CYP2C8 P10632 1/20 0.53
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12000614 0.92 S1PR1 (0.65) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL21351518 0.88 S1PR1 (0.67) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1813959 0.88 S1PR1 (0.67) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL12076028 0.88 S1PR1 (0.77) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1814365 0.86 S1PR1 (0.74) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1815061 0.84 S1PR1 (0.65) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1805834 0.84 S1PR1 (0.68) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1815074 0.84 S1PR1 (0.66) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1815683 0.83 S1PR1 (0.84) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL12000613 0.83 S1PR1 (0.64) S1PR1S1PR3CYP3A4CYP2C8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2592071-B1 Tricyclic heterocyclic compounds BRISTOL MYERS SQUIBB CO (US) 2019-09-18 EP claimed
US-9216972-B2 Tricyclic heterocyclic compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2015-12-22 US claimed