SCHEMBL173539

SCHEMBL173539

CNC(=O)c1ccc(Nc2ncnc3cc(OC)c(NC(=O)[C@@H]4CCCN4C(=O)[C@@H](NC[C@H](C)NC)C(C)(C)C)cc23)cc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.60
CYP2C9 P11712 2/20 0.60
CYP2C19 P33261 1/20 0.60
XIAP P98170 1/20 0.60
KDR P35968 10/20 0.44
EGFR P00533 5/20 0.44
ERBB2 P04626 5/20 0.44
RAF1 P04049 2/20 0.44
FGFR2 P21802 2/20 0.44
FLT4 P35916 2/20 0.44
TEK Q02763 2/20 0.44
ABL1 P00519 1/20 0.44
LCK P06239 1/20 0.44
RET P07949 1/20 0.44
SRC P12931 1/20 0.44
FLT1 P17948 1/20 0.44
ERBB4 Q15303 3/20 0.44
JAK3 P52333 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173674 0.92 CYP3A4 (0.61) CYP3A4CYP2C9CYP2C19XIAPKDR
Hydrochloric Acid SCHEMBL168317 0.92 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19XIAPKDR
Hydrochloric Acid SCHEMBL170945 0.91 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19XIAPKDR
SCHEMBL174167 0.90 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19XIAPKDR
SCHEMBL173786 0.90 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19XIAPKDR
Hydrochloric Acid SCHEMBL173396 0.89 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19XIAPKDR
SCHEMBL15050426 0.89 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19XIAPKDR
SCHEMBL157401 0.89 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19XIAPKDR
SCHEMBL15050425 0.89 CYP3A4 (0.76) CYP3A4CYP2C9CYP2C19XIAPKDR
Hydrochloric Acid SCHEMBL170502 0.89 CYP3A4 (0.58) CYP3A4CYP2C9CYP2C19XIAPKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611797-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS Hanmi Science Co., Ltd. (KR) 2013-07-10 EP disclosed
WO-2012030160-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS HANMI HOLDINGS CO., LTD. (KR) 2012-03-08 WO disclosed