SCHEMBL17377352

SCHEMBL17377352

NC(=NO)c1ccc(Nc2nnc(-c3ccc(Cl)cc3)o2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.63
ACHE P22303 1/20 0.50
QPCT Q16769 1/20 0.49
SPHK2 Q9NRA0 1/20 0.49
HDAC6 Q9UBN7 1/20 0.48
HDAC1 Q13547 1/20 0.47
KDM4E B2RXH2 2/20 0.47
ADCY1 Q08828 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
ATR Q13535 1/20 0.46
LMNA P02545 1/20 0.46
ALOX15 P16050 1/20 0.46
ALOX12 P18054 1/20 0.46
CXCR5 P32302 1/20 0.46
APLNR P35414 1/20 0.46
OPRK1 P41145 1/20 0.46
CCR6 P51684 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PTGS2 P35354 1/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17377350 1.00 GSK3B (0.63) GSK3BACHEQPCTSPHK2HDAC6
SCHEMBL19077663 0.90 GSK3B (0.60) GSK3BACHEQPCTSPHK2HDAC6
SCHEMBL17377394 0.85 NPC1 (0.53) KDM4EADCY1SMN1; SMN2LMNAPTGS2
SCHEMBL17377396 0.85 NPC1 (0.53) KDM4EADCY1SMN1; SMN2LMNAPTGS2
SCHEMBL17377364 0.85 GSK3B (0.62) GSK3BACHEQPCTSPHK2HDAC6
SCHEMBL17383549 0.85 GSK3B (0.62) GSK3BACHEQPCTSPHK2HDAC6
Hydrochloric Acid SCHEMBL17377355 0.84 GSK3B (0.61) GSK3BACHEQPCTSPHK2HDAC6
SCHEMBL3532271 0.80 SPHK2 (0.74) GSK3BACHEQPCTSPHK2HDAC1
SCHEMBL17377392 0.80 SPHK2 (0.74) GSK3BACHEQPCTSPHK2HDAC1
SCHEMBL17377351 0.79 GSK3B (0.61) GSK3BACHEQPCTSPHK2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9828351-B2 Enzyme interacting agents MONASH UNIVERSITY (AU) 2017-11-28 US disclosed
US-20170190698-A1 ENZYME INTERACTING AGENTS CENTRAL ADELAIDE LOCAL HEALTH NETWORK INCORPORATED (AU) 2017-07-06 US disclosed
EP-3160949-A1 ENZYME INTERACTING AGENTS Monash University (AU) 2017-05-03 EP disclosed
WO-2015196258-A1 ENZYME INTERACTING AGENTS MONASH UNIVERSITY (AU) 2015-12-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170190698-A1 ENZYME INTERACTING AGENTS SMPD1, SMPD2, ASAH1 GSK3B 3195/4885ACHE 430/4885QPCT 980/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.