SCHEMBL17387451

SCHEMBL17387451

O=C(c1ccc(F)cc1)N1CCC(N2C[C](n3cc(-c4ncnc5[nH]ccc45)cn3)C2)CC1

nearest known ligand 0.67

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 20/20 0.67
JAK1 P23458 10/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17957113 0.93 JAK2 (0.67) JAK2JAK1
SCHEMBL14563474 0.92 JAK2 (0.66) JAK2JAK1
SCHEMBL17957104 0.91 JAK2 (0.68) JAK2JAK1
SCHEMBL17957103 0.91 JAK2 (0.67) JAK2JAK1
SCHEMBL17957100 0.91 JAK2 (0.68) JAK2JAK1
SCHEMBL14563783 0.90 JAK2 (0.68) JAK2JAK1
SCHEMBL17387467 0.90 JAK2 (0.69) JAK2JAK1
SCHEMBL14563463 0.90 JAK2 (0.69) JAK2JAK1
SCHEMBL14563414 0.89 JAK2 (0.69) JAK2JAK1
SCHEMBL14563583 0.89 JAK2 (0.69) JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050882-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS Incyte Holdings Corporation (US) 2016-08-03 EP claimed
EP-2545045-B1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS INCYTE HOLDINGS CORP (US) 2016-01-06 EP claimed
EP-3050882-A1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS Incyte Holdings Corporation (US) 2016-08-03 EP disclosed
EP-2545045-B1 PIPERIDIN-4-YL AZETIDINE DERIVATIVES AS JAK1 INHIBITORS INCYTE HOLDINGS CORP (US) 2016-01-06 EP disclosed